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نالمكسون (بالإنجليزية: Nalmexone) هو مسكّن ألم قوي من فئة الأفيونيات. يعمل نالمكسون بشكل مباشر على الجهاز العصبي المركزي لتقليل الشعور بالألم. يمكن استخدامه لكل من الألم الحاد والألم المزمن.
, Nalmexone (INN) (code names EN-1620A, UM-5 … Nalmexone (INN) (code names EN-1620A, UM-592), or nalmexone hydrochloride (USAN), is a semisynthetic, opioid partial agonist or mixed agonist-antagonist with both analgesic and narcotic antagonist properties that was never marketed. In clinical studies it was found to have comparable analgesic efficacy to morphine, though with several-fold reduced potency. In addition, nalmexone's side effects, the most common of which were sleepiness and sweating, were reported to be similar to those of morphine, albeit with a noticeably higher degree of incidence.h a noticeably higher degree of incidence.
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rdfs:comment |
Nalmexone (INN) (code names EN-1620A, UM-5 … Nalmexone (INN) (code names EN-1620A, UM-592), or nalmexone hydrochloride (USAN), is a semisynthetic, opioid partial agonist or mixed agonist-antagonist with both analgesic and narcotic antagonist properties that was never marketed. In clinical studies it was found to have comparable analgesic efficacy to morphine, though with several-fold reduced potency. In addition, nalmexone's side effects, the most common of which were sleepiness and sweating, were reported to be similar to those of morphine, albeit with a noticeably higher degree of incidence.h a noticeably higher degree of incidence.
, نالمكسون (بالإنجليزية: Nalmexone) هو مسكّن ألم قوي من فئة الأفيونيات. يعمل نالمكسون بشكل مباشر على الجهاز العصبي المركزي لتقليل الشعور بالألم. يمكن استخدامه لكل من الألم الحاد والألم المزمن.
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rdfs:label |
نالمكسون
, Nalmexone
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